Eskandar ALIPOUR, Asghar DAVOOD, Abbas SHAFIEE

5675

Efficcient synthesis of imidazole derivatives: An important synthon for the preparation of biologically active compounds

Efficcient synthesis of imidazole derivatives: An important synthon for the preparation of biologically active compounds

4(5)-Chloro-imidazole-5(4)-carboxaldehyde derivatives are important precursors for the preparation of biologically active compounds. We developed a simple, novel, and efficient method for the synthesis of these compounds. The chemistry described is amenable to large-scale use and is flexible enough to allow the preparation of analogs.
PDF

___

  • 1.A. Davood, G. Khodarahmi, E. Alipour, A. Dehpour, M. Amini and A. Shafiee, Boll. Chim. Farm- 140, 381-386 (2001).
  • 2.G.J. Griffiths, M.B. Hauck, R. Imwinkelried, J. Kohr, C.A. Rotten and G.C. Stucky, J. Org. Chem. 64, 8084-8089 (1999).
  • 3.T. Murai, T. Saak, S. Satous, S. Mura, T. Takashige, Y. Ikeda and N. Kane, Eur. Patent 0611, 758, Chem. Abstr. 121, 230770x (1994).
  • 4.C.H. Zhou, Z.C. Liu., R.G. Xie and H.M. Zhao, Chin. Chem. Lett. 8, 21-24 (1997).
  • 5.S.P Watson, Synthetic Commun. 22, 2971-2977 (1992).
  • 6.A. Davood, N. Mansouri, A.R. Dehpour, H. Shafaroudi, E. Alipour and A. Shafiee. Archiv Der Pharmazie,339, 299-304 (2006).
  • 7.R. Weidenhagen and R. Herrmann, Ber. 68, 1953-1961 (1935).
  • 8.A.R. Katrizky, Handbook of Heterocyclic Chemistry, 1st ed. pp. 307-311 Pergamon Press, Oxford, 1985.
Turkish Journal of Chemistry-Cover
  • ISSN: 1300-0527
  • Yayın Aralığı: 6
  • Yayıncı: TÜBİTAK
Arşiv
Sayıdaki Diğer Makaleler

Synthesis of some new 4-oxo-4H chromene derivatives bearing nitrogen heterocyclic systems as antifungal agents

El- Sayed Tarik ALI, Abdel- Aghfaar Salah ABDEL-AZIZ, Metwali Hafez EL-SHAAER, Ismail Faten HANAFY, Zaky Ali EL-FAUOMY

Efficcient synthesis of imidazole derivatives: An important synthon for the preparation of biologically active compounds

Eskandar ALIPOUR, Asghar DAVOOD, Abbas SHAFIEE

Cyanoacetamide Derivatives as Synthons in Heterocyclic Synthesis

Ahmed Ali FADDA, Samir BONDOCK, Ramy RABIE

Characterization and Antimicrobial Activity of Organotin(IV) Complexes of 2-[(2´,6´-diethylphenylamido)]benzoates and 3-[(2´,6´-diethylphenylamido)]propanoates

Saira SHAHZADI, Khadija SHAHID, Saqib ALI, Mohammad BAKHTIAR

Efficient Synthesis of Imidazole Derivatives: An Important Synthon for the Preparation of Biologically Active Compounds

Asghar DAVOOD, Eskandar ALIPOUR, Abbas SHAFIEE

Synthesis and Characterization of Novel Polyamide and Polyhydrazides Based on the 6,6´-disubstituted-2,2´-bipyridine

Abdurrahman ŞENGÜL, Hülya ARSLAN

A Hydrogen Ion-Selective Poly(Vinyl Chloride) Membrane Electrode Based on Calix[4]arene as a Perchlorate Ion-Selective Electrode

Esin CANEL, Sevcan ERDEN, Ayça DEMİREL ÖZEL, Sahahabuddin MEMON

Synthesis and Swelling Behavior of Starch-Poly (Sodium Acrylate-co-Acrylamide) Superabsorbent Hydrogel

Mohammad SADEGHI, Hossein HOSSEINZADEH

Characterization and antimicrobial activity of organotin (IV) complexes of 2-(2',6'-diethylphenylamido) benzoates and 3-(2',6'-diethylphenylamido) propanoates

Mohammad BAKHTIAR, Khadija SHAHID, Saqib ALI, Saira SHAHZADI

Behaviour of Salicylaldehyde and Some of Its Derivatives in the Biginelli Reaction for the Preparation of Aryl Tetrahydropyrimidines

Eman Moustafa Hassan ABBAS, Shadia Mahmoud ABDALLAH